Home Tools
Log in
Cart

Search Result

Search Results for " tachykinin receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T7633 Senktide Neurokinin receptor
Senktide is an agonist of tachykinin NK3 receptor.
T7209 Maropitant Neurokinin receptor
Maropitant is a selective neurokinin (NK1) receptor antagonist.
TP1087 Substance P Neurokinin P Endogenous Metabolite , Neurokinin receptor
Substance P (Neurokinin P) (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) member of the tachykinin neuropeptide family.
TP1572 GR-73632 Neurokinin receptor
Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).
T38144 Elinzanetant Neurokinin receptor
Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.
T15278 Fezolinetant ESN-364 Neurokinin receptor
Fezolinetant (ESN-364) is an antagonist of the neurokinin 3 receptor (NK3R). It is used for the treatment of menopausal hot flushes.
T23316 SB 218795 Neurokinin receptor
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
T7549 Talnetant SB 223412 Neurokinin receptor
Talnetant (SB 223412) is a selective, competitive, brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission
T16849 SB-222200 Neurokinin receptor
SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
T8235 L-732138 Neurokinin receptor
L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)
TP1883 [Lys5,MeLeu9,Nle10]-NKA(4-10) Neurokinin receptor
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
T17156 Tradipitant VLY-686,LY686017 Neurokinin receptor
Tradipitant (VLY-686) is an antagonist of neurokinin-1.
T7554 Substance P (7-11) Substance P 7-11(TFA) Others , Neurokinin receptor
Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .
T6905 Netupitant Ro 67-31898/000,CID 6451149 Neurokinin receptor
Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).
T3716 Rolapitant SCH619734 Neurokinin receptor
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ...
TP1008 Neurokinin A α-Neurokinin,Substance K,Neuromedin L Neurokinin receptor
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.
T1743 Aprepitant MK-869,MK-0869,L-754030,Aprepitant` HIV Protease , Antibacterial , Antibiotic , Neurokinin receptor
Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist. The mechanism of action of aprepitant is as a Neurokinin 1 Antagonist, and Cytochrome P450 3A4 Inhibitor, and Cytochrome P450 2C9 Inducer, and C...
T13306L Vapreotide acetate RC-160 acetate,BMY-41606 acetate Neurokinin receptor
Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).
T3034 Eprazinone dihydrochloride Resplen,Mucitux,Eftapan,NSC 317935,Eprazinone 2HCl Others , Neurokinin receptor
Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.
T1790 Fosaprepitant dimeglumine L785298,MK-0517,Fosaprepitant dimeglumine salt Neurokinin receptor
Fosaprepitant dimeglumine (MK-0517) is the dimeglumine salt form of fosaprepitant, the water-soluble, N-phosphorylated prodrug of aprepitant, with antiemetic activity. Upon intravenous administration and rapid conversion...

Compounds

Senktide
T7633
Synonym:
Target: Neurokinin receptor
Maropitant
T7209
Synonym:
Target: Neurokinin receptor
Substance P
TP1087
Synonym: Neurokinin P
Target: Endogenous Metabolite, Neurokinin receptor
GR-73632
TP1572
Synonym:
Target: Neurokinin receptor
Elinzanetant
T38144
Synonym:
Target: Neurokinin receptor
Fezolinetant
T15278
Synonym: ESN-364
Target: Neurokinin receptor
SB 218795
T23316
Synonym:
Target: Neurokinin receptor
Talnetant
T7549
Synonym: SB 223412
Target: Neurokinin receptor
SB-222200
T16849
Synonym:
Target: Neurokinin receptor
L-732138
T8235
Synonym:
Target: Neurokinin receptor
[Lys5,MeLeu9,Nle10]-NKA(4-10)
TP1883
Synonym:
Target: Neurokinin receptor
Tradipitant
T17156
Synonym: VLY-686,LY686017
Target: Neurokinin receptor
Substance P (7-11)
T7554
Synonym: Substance P 7-11(TFA)
Target: Others, Neurokinin receptor
Netupitant
T6905
Synonym: Ro 67-31898/000,CID 6451149
Target: Neurokinin receptor
Rolapitant
T3716
Synonym: SCH619734
Target: Neurokinin receptor
Neurokinin A
TP1008
Synonym: α-Neurokinin,Substance K,Neuromedin L
Target: Neurokinin receptor
Aprepitant
T1743
Synonym: MK-869,MK-0869,L-754030,Aprepitant`
Target: HIV Protease, Antibacterial, Antibiotic, Neurokinin receptor
Vapreotide acetate
T13306L
Synonym: RC-160 acetate,BMY-41606 acetate
Target: Neurokinin receptor
Eprazinone dihydrochloride
T3034
Synonym: Resplen,Mucitux,Eftapan,NSC 317935,Eprazinone 2HCl
Target: Others, Neurokinin receptor
Fosaprepitant dimeglumine
T1790
Synonym: L785298,MK-0517,Fosaprepitant dimeglumine salt
Target: Neurokinin receptor
1 2 3 4 5
TargetMol